Development of an oxazole conjunctive reagent and application to the total synthesis of siphonazoles.

نویسندگان

  • Jianmin Zhang
  • Elena A Polishchuk
  • Jie Chen
  • Marco A Ciufolini
چکیده

The preparation of 4-carbethoxy-5-methyl-2-(phenylsulfonyl)methyloxazole and its use in the elaboration of more complex oxazoles are described. A total synthesis of the unique natural products siphonazoles A and B, illustrates an application of this building block. A discussion of the biological activity of the siphonazoles is also presented.

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عنوان ژورنال:
  • The Journal of organic chemistry

دوره 74 23  شماره 

صفحات  -

تاریخ انتشار 2009